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Derniers dépôts
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Nathan Picois, Lizeth Bodero, Pierre T Milbeo, Thierry Brigaud, Grégory Chaume. Bimodal use of chiral α‐Trifluoromethylalanine in Aib Foldamers: study of the position impact towards the helical screw‐sense preference. Chemistry - A European Journal, In press, ⟨10.1002/chem.202400540⟩. ⟨hal-04516499⟩
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Julia Kaffy, Dimitri Brinet, Jean-Louis Soulier, Isabelle Correia, Nicolo Tonali, et al.. Designed Glycopeptidomimetics Disrupt Protein–Protein Interactions Mediating Amyloid β-Peptide Aggregation and Restore Neuroblastoma Cell Viability. Journal of Medicinal Chemistry, 2016, 59 (5), pp.2025-2040. ⟨10.1021/acs.jmedchem.5b01629⟩. ⟨hal-02467871⟩
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Doumet Georges Helou, A. Mauras, Francois Fasquelle, J. S. Lanza, P. M. Loiseau, et al.. Intranasal vaccine from whole Leishmania donovani antigens provides protection and induces specific immune response against visceral leishmaniasis.. PLoS Neglected Tropical Diseases, 2021, PLoS Neglected Tropical Diseases, 15, pp.e0009627. ⟨10.1371/journal.pntd.0009627⟩. ⟨hal-04482585⟩
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Nicolas Duchemin, Adam Skiredj, Justine Mansot, Karine Leblanc, Jean-Jacques Vasseur, et al.. DNA-Templated [2+2] Photocycloaddition: A Straightforward Entry into the Aplysinopsin Family of Natural Products. Angewandte Chemie International Edition, 2018, 57 (36), pp.11786-11791. ⟨10.1002/anie.201806357⟩. ⟨hal-02197152⟩
Mots-clés
C-nucleoside
Antimicrobial activity
Cytotoxicity
Fluor
Aggregation
Annulations
Antiviral
Chemistry
Ribavirin
Alkaloids
Biological activity
Mass spectrometry
Acetogenin
Glycosylation
Buchwald-Hartwig-Migita coupling
Enynes
Amyloid
Alkynylation
Biomimetic synthesis
Force-field
Sodium iodide
Benzils
Halogenation
Chemical diversity
Michael addition
Annonacin
Human
Hair
Antimalarial
Controlled study
Conformational analysis
Peptidomimetics
Amyloïde
Biosynthesis
Capillary electrophoresis
Hydrostannation
Antimitotic
Chalcones
Archéométrie des matières colorantes
Conformational ensemble
Biotransformation
Cancer
Molecular dynamics
ACL
Combretastatin A-4
Palladium
Cyclization
Ilimaquinone
Chitosan
NMR
CXCR4
Synthetic methods
Benzofuran
Autoimmune diseases
Binding
IsoCA-4
Environmental neurotoxin
Apoptosis
Dereplication
Fluorescence
Tubulin
Constrained amino acids
Aldehydes
Molecular networking
Fluorine
Leishmania
DMSO
Foldamers
Circular dichroism
Carbohydrates
Leishmaniasis
Catalysis
Benthic cyanobacteria
Biosynthèse
Copper
Alteration
High-resolution mass spectrometry
Article
Autoanticorps
Binding site
Amphidinolide
Natural products
5-HT 4 receptor
Fluorinated peptides
Coupling
Heterocycles
Crystallography
Autoantibodies
Molecular modeling
Alkynes
Antileishmanial
Glycosides
Annonaceae
Alkyne
Thiosugars
Pigments
Peptidomimétiques
Peptides
Asymmetric synthesis
Alpha-synuclein